HRH4_HUMAN
General information
| Gene Name | HRH4 |
| Family | Histamine type 4 |
| GPCRDB | HRH4_HUMAN |
| UniProt | Q9H3N8 |
| IUPHAR | 2967 |
| Entrez Gene | 59340 |
| KEGG | hsa:59340 |
| Sequence | HRH4_HUMAN.fasta |
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Binding information
Agonist
|
|
Name(s) |
2-methylhistamine |
| PubChem Compound | 91613 | |
| Formula | C6 H11 N3 | |
| Mol. Wt. | 125.095 | |
| Cas No. | 34392-54-6 | |
| KEGG | ||
| ChEBI | ||
| DrugBank | ||
| Struct. file | L000064.mol L000064.kegg | |
| Activity | Full Agonist | |
| Reference | PMID:16432504 PMID:15947036 | |
|
|
Name(s) |
4-methylhistamine |
| PubChem Compound | 37463 | |
| Formula | C6 H11 N3 | |
| Mol. Wt. | 125.095 | |
| Cas No. | 36376-47-3 36507-31-0 | |
| KEGG | ||
| ChEBI | ||
| DrugBank | ||
| Struct. file | L000072.mol L000072.kegg | |
| Activity | Full Agonist | |
| Reference | PMID:16432504 PMID:15947036 | |
|
|
Name(s) |
Dimaprit |
| PubChem Compound | 3077 | |
| Formula | C6 H15 N3 S | |
| Mol. Wt. | 161.099 | |
| Cas No. | 23256-33-9 65119-89-3 | |
| KEGG | ||
| ChEBI | ||
| DrugBank | ||
| Struct. file | L000225.mol L000225.kegg | |
| Activity | Full Agonist | |
| Reference | PMID:11179434 PMID:11179436 PMID:15947036 PMID:11181941 | |
|
|
Name(s) |
Histamine |
| PubChem Compound | 774 | |
| Formula | C5 H9 N3 | |
| Mol. Wt. | 111.080 | |
| Cas No. | 51-45-6 56-92-8 | |
| KEGG | C00388 | |
| ChEBI | 18295 | |
| DrugBank | EXPT01785 | |
| Struct. file | L000292.mol L000292.kegg | |
| Activity | Full Agonist | |
| Reference | PMID:11561071 PMID:11179434 PMID:16432504 PMID:11179436 PMID:15947036 PMID:11181941 PMID:15454206 PMID:11179435 PMID:10973974 PMID:15033391 | |
|
|
Name(s) |
imetit |
| PubChem Compound | 3692 | |
| Formula | C6 H10 N4 S | |
| Mol. Wt. | 170.063 | |
| Cas No. | 102203-18-9 | |
| KEGG | ||
| ChEBI | ||
| DrugBank | ||
| Struct. file | L000309.mol L000309.kegg | |
| Activity | Full Agonist | |
| Reference | PMID:11561071 PMID:11179434 PMID:11179436 PMID:11181941 | |
|
|
Name(s) |
4-(1H-imidazol-4-ylmethyl)piperidine |
| PubChem Compound | 3035842 | |
| Formula | C9 H15 N3 | |
| Mol. Wt. | 165.127 | |
| Cas No. | 151070-83-6 | |
| KEGG | ||
| ChEBI | ||
| DrugBank | ||
| Struct. file | L000311.mol L000311.kegg | |
| Activity | Full Agonist | |
| Reference | PMID:11179434 PMID:11179436 PMID:14640553 | |
|
|
Name(s) |
Impromidine |
| PubChem Compound | 41376 | |
| Formula | C14 H23 N7 S | |
| Mol. Wt. | 321.173 | |
| Cas No. | 55273-05-7 65573-02-6 | |
| KEGG | ||
| ChEBI | ||
| DrugBank | ||
| Struct. file | L000313.mol L000313.kegg | |
| Activity | Partial Agonist | |
| Reference | PMID:11179434 PMID:15947036 PMID:12954048 | |
|
|
Name(s) |
N-methylhistamine |
| PubChem Compound | 912 | |
| Formula | C6 H11 N3 | |
| Mol. Wt. | 125.095 | |
| Cas No. | 673-50-7 | |
| KEGG | ||
| ChEBI | ||
| DrugBank | ||
| Struct. file | L000451.mol L000451.kegg | |
| Activity | Full Agonist | |
| Reference | PMID:11179436 PMID:11181941 | |
|
|
Name(s) |
N-methylhistamine |
| PubChem Compound | 912 | |
| Formula | C6 H11 N3 | |
| Mol. Wt. | 125.095 | |
| Cas No. | 673-50-7 | |
| KEGG | ||
| ChEBI | ||
| DrugBank | ||
| Struct. file | L000451.mol L000451.kegg | |
| Activity | Full Agonist | |
| Reference | PMID:11179434 | |
|
|
Name(s) |
alpha-methylhistamine |
| PubChem Compound | 3615 | |
| Formula | C6 H11 N3 | |
| Mol. Wt. | 125.095 | |
| Cas No. | 6986-90-9 | |
| KEGG | ||
| ChEBI | ||
| DrugBank | ||
| Struct. file | L000527.mol L000527.kegg | |
| Activity | Full Agonist | |
| Reference | PMID:11179434 | |